Publications

For a free electronic reprint of any Burke Group publication, please email Ramona Rudzinski at ramonar@illinois.edu

98. Stereospecific Csp3 Suzuki-Miyaura Cross-Coupling That Evades b-Oxygen Elimination, Antonio J. LaPorte, Yao Shi, Jason E. Hein, and Martin D. Burke, ACS Catal. 2022, 12, 10905-10912. DOI: https://doi.org/10.1021/acscatal.2c03245

97. A small molecule redistributes iron in ferroportin-deficient mice and patient-derived primary macrophages, Stella Ekaputria, Eun-Kyung Choi, Manuela Sabelli, Luisa Aring, Kelsie J. Green, JuOae Chang, Kai Bao, Hak Soo Choi, Shigeki Iwase, Jonghan Kim, Elena Corradini, Antonello Pietrangelo, Martin D. Burke and Young Ah Seo Natl. Acad. Sci. U.S.A. 2022, 119, e2121400119 https://doi.org/10.1073/pnas.2121400119

96. Targeting fungal membrane homeostasis with imidazopyrazoindoles impairs azole resistance and biofilm formation, Nicole M. Revie, Kali R. Iyer, Michelle E. Maxson, Jiabao Zhang, Su Yan, Caroline M. Fernandes, Kirsten J. Meyer, Xuefei Chen, Iwona Skulska, Meea Fogal, Hiram Sanchez, Saif Hossain, Sheena Li, Yoko Yashiroda, Hiroyuki Hirano, Minoru Yoshida, Hiroyuki Osada, Charles Boone, Rebecca S. Shapiro, David R. Andes, Gerard D. Wright, Justin R. Nodwell, Maurizio Del Poeta, Martin D. Burke, Luke Whitesell, Nicole Robbins & Leah E. Cowen Nat Commun13, 3634, 2022 https://doi.org/10.1038/s41467-022-31308-1

95. MIDA Anhydride and Reaction with Boronic Acids,Aidan M. Kelly, Peng-Jui Chen, Jenna Klubnick, Daniel J. Blair, and Martin D. Burke Org. Synth.202299, 92 DOI: 10.15227/orgsyn.099.0092

94. Digitizing Chemical Synthesis in 3D Printed Reactionware, Andrius Bubliauskas, Daniel J. Blair, Henry Powell-Davies, Philip J. Kitson, Martin D. Burke, Leroy Cronin Acknow, Angew. Chem. Int. Ed.2022, e202116108; Angew. Chem.2022, e202116108

93. Mitigation of SARS-CoV-2 Transmission at a Large Public University, Diana Rose E. Ranoa, Robin L. Holland, Fadi G. Alnaji, Kelsie J. Green, Leyi Wang, Richard L. Fredrickson, Tong Wang, George N. Wong, Johnny Uelmen, Sergei Maslov, Ahmed Elbanna, Zachary J. Weiner, Alexei V. Tkachenko, Hantao Zhang, Zhiru Liu, Sanjay J. Patel, John M. Paul, Nickolas P. Vance, Joseph G. Gulick, Sandeep Puthanveetil Satheesan, Isaac J. Galvan, Andrew Miller, Joseph Grohens, Todd J. Nelson, Mary P. Stevens, P. Mark Hennessy, Robert C. Parker Jr, Edward Santos, Charles Brackett, Julie D. Steinman, Melvin R. Fenner Jr, Kirstin Dohrer, Kraig Wagenecht, Michael DeLorenzo, Laura Wilhelm-Barr, Brian R. Brauer, Catherine Best-Popescu, Gary Durack, Nathan Wetter, David M. Kranz,  Jessica Breitbarth, Charlie Simpson, Julie A. Pryde, Robin N. Kaler, Chris Harris, Allison C. Vance, Jodi L. Silotto, Mark Johnson, Enrique Valera, Patricia K. Anton, Lowa Mwilambwe,  Stephen P. Bryan, Deborah S. Stone, Danita B. Young, Wanda E. Ward, John Lantz, John A. Vozenilek, Rashid Bashir, Jeffrey S. Moore, Mayank Garg, Julian C. Cooper, Gillian Snyder,  Michelle H. Lore, Dustin L. Yocum, Neal J. Cohen, Jan E. Novakofski, Melanie J. Loots, Randy L. Ballard, Mark Band, Kayla M. Banks, Joseph D. Barnes, Iuliana Bentea, Jessica Black,  Jeremy Busch, Hannah Christensen, Abigail Conte, Madison Conte, Michael Curry, Jennifer Eardley, April Edwards, Therese Eggett, Judes Fleurimont, Delaney Foster, Bruce W. Fouke,  Nicholas Gallagher, Nicole Gastala, Scott A. Genung,  Declan Glueck, Brittani Gray,  Andrew Greta, Robert M. Healy, Ashley Hetrick, Arianna A Holterman, Nahed Ismail, Ian Jasenof, Patrick Kelly, Aaron Kielbasa, Teresa Kiesel, Lorenzo M. Kindle, Rhonda L. Lipking, Yukari C. Manabe, Jade Mayes, Reubin McGuffin, Kenton G. McHenry, Agha Mirza, Jada Moseley, Heba H. Mostafa, Melody Mumford,   Kathleen Munoz, Arika D. Murray, Moira Nolan, Nil A. Parikh, Andrew Pekosz, Janna Pflugmacher, Janise M. Phillips, Collin Pitts, Mark C. Potter, James Quisenberry, Janelle Rear, Matthew L. Robinson, Edith Rosillo, Leslie N. Rye, MaryEllen Sherwood, Anna Simon, Jamie M. Singson, Carly Skadden, Tina H. Skelton, Charlie Smith, Mary Stech, Ryan Thomas, Matthew A. Tomaszewski, Erika A. Tyburski, Scott Vanwingerden, Evette Vlach, Ronald S. Watkins, Karriem Watson, Karen C. White, Timothy L. Killeen, Robert J. Jones, Andreas C. Cangellaris, Susan A. Martinis, Awais Vaid, Christopher B. Brooke, Joseph T. Walsh,  William C. Sullivan, Rebecca L. Smith, Nigel D. Goldenfeld, Timothy M. Fan, Paul J. Hergenrother, Martin D. Burke Nat Commun 13, 3207, 2022. https://doi.org/10.1038/s41467-022-30833-3

92. Using automated synthesis to understand the role of side chains on molecular charge transport, Songsong Li, Edward R. Jira, Nicholas H. Angello, Jialing Li, Hao Yu, Jeffrey S. Moore, Ying Diao, Martin D. Burke, and Charles M. Schroeder Nat Commun13, 2102. 2022,https://doi.org/10.1038/s41467-022-29796-2

91. Automated iterative Csp3-C bond formation, Daniel J. Blair, Sriyankari Chitti, Melanie Trobe, David M. Kostyra, Hannah M. S. Haley, Richard L. Hansen, Steve G. Ballmer, Toby J. Woods, Wesley Wang, Vikram Mubayi, Michael J. Schmidt, Robert W. Pipal, Greg. F. Morehouse, Andrea M. E. Palazzolo Ray, Danielle L. Gray, Adrian L. Gill & Martin D. Burke Nature 2022, https://doi.org/10.1038/s41586-022-04491-w

90. A Materials Acceleration Platform for Organic Laser Discovery, Tony C. Wu, Andrés Aguilar Granda, Kazuhiro Hotta, Sahar Alasvand Yazdani, Robert Pollice, Jenya Vestfrid, Han Hao, Cyrille Lavigne, Martin Seifrid, Nicholas H. Angello, Fatima Bencheikh, Jason E. Hein, Martin D. Burke, Chihaya Adachi, Alán Aspuru-Guzik ChemRxiv. Cambridge: Cambridge Open Engage; 2022 DOI 10.26434/chemrxiv-2022-9zm65

89. Automated Synthesis for Single-Molecule Electronics, Edward R. Jira, Songsong Li, Nicholas H. Angello, Jialing Li, Jeffrey S. Moore, Martin D. Burke, Charles M. Schroeder Bulletin of the American Physical Society, 2022

88. Machine Learning May Sometimes Simply Capture Literature Popularity Trends: A Case Study of Heterocyclic Suzuki-Miyaura Coupling, Wiktor Beker, Rafał Roszak, Agnieszka Wołos, Nicholas H. Angello, Vandana Rathore, Martin D. Burke, and Bartosz A. Grzybowski J. Am. Chem. Soc.2022, 144, 11, 4819–4827 https://doi.org/10.1021/jacs.1c12005

87. Iterations from the chemical cosmos, Danielle C. Loving and Martin D. Burke Nature Synth1, 11–12 2022, https://doi.org/10.1038/s44160-021-00014-z

86. Validation of a molecular assay to detect SARS-CoV-2 in saliva, Janet L. Pitman, Arthur J. Morris, Stephen Grice, Joseph T. Walsh, Leyi Wang, Martin D. Burke, Amanda Dixon-McIver The New Zealand Medical Journal, Vol 134 No 1547: 17 2021

85. Chemical-Reaction-Aware Molecule Representation Learning, Hongwei Wang, Weijiang Li, Xiaomeng Jin, Kyunghyun Cho, Heng Ji, Jiawei Han, Martin D. Burke arXiv2021

84. Hybrid Amphotericin B derivatives with reduced toxicity, Martin D. Burke, Anuj Khandelwal, Jiabao Zhang, Anna SantaMaria, US Patent 11,198,705. 2021

83. Fungicidal Amphotericin B Sponges are Assemblies of Staggered Asymmetric Homodimers Encasing Large Void Volumes, Agnieszka Lewandowska, Corinne P. Soutar, Alexander I. Greenwood, Evgeny Nimerovsky, Ashley M. De Lio, Jordan T. Holler, Grant S. Hisao, Anuj Khandelwal, Jiabao Zhang, Anna M. SantaMaria, Charles D. Schwieters, Taras V. Pogorelov, Martin D. Burke & Chad M. Rienstra Nature Structural & Molecular Biology 2021, 12, 972-981 DOI: 10.1038/s41594-021-00685-4

82. Chemical-Reaction-Aware Molecule Representation Learning, Hongwei Wang, Weijiang Li, Xiaomeng Jin, Kyunghyun Cho, Heng Ji, Jiawei Han, Martin D. Burke arXiv2021

81. Transition between Nonresonant and Resonant Charge Transport in Molecular Junctions, Songsong Li, Hao Yu, Jialing Li, Nicholas Angello, Edward R. Jira, Bo Li, Martin D. Burke, Jeffrey S. Moore, and Charles M. Schroeder Nano Letters 202121(19), 8340-8347 DOI: 10.1021/acs.nanolett.1c02915

80. Well-Tolerated Amphotericin B Derivatives That Effectively Treat Visceral Leishmaniasis, Christelle Morelle, Angana Mukherjee, Jiabao Zhang, Fereshteh Fani, Anuj Khandelwal, Hélène Gingras, Jocelyn Trottier, Olivier Barbier, Philippe Leprohon, Martin D. Burke, and Marc Ouellette ACS Infectious Diseases 2021, 7(8), 2472-2482 DOI: 10.1021/acsinfecdis.1c00245

79. Sterol Sponge Mechanism Is Conserved for Glycosylated Polyene Macrolides, Xiaorui Guo, Jiabao Zhang, Xinyi Li, Emily Xiao, Justin D. Lange, Chad M. Rienstra, Martin D. Burke, and Douglas A. Mitchell ACS Central Science20217 (5), 781-791 DOI: 10.1021/acscentsci.1c00148

78. Amphotericin B induces epithelial voltage responses in people with cystic fibrosis Rajeev S. Chorghade, Bo Ram Kim, Janice L. Launspach, Philip H. Karp, Michael J. Welsh and Martin D. Burke Journal of Cystic Fibrosis 2020,7 (5), 781-791 DOI: 10.1016/j.jcf.2020.11.01

77. COVID-19 Testing Strategies for Colleges and Universities National Academies of Sciences, Engineering, and Medicine.’ Washington, DC: The National Academies Press, 2020

76. Saliva-Based Molecular Testing for SARS-CoV-2 that Bypasses RNA Extraction Diana Rose E. Ranoa, Robin L. Holland, Fadi G. Alnaji, Kelsie J. Green, Leyi Wang, Christopher Byron Brooke, Martin D. Burke, Timothy M. Fan, Paul Hergenrother Cold Spring Harbor Laboratory Press, 2020 DOI: 10.1101/2020.06.18.159434v1

75. Derivatives of Amphotericin B, Martin D. Burke, Arun P. Thottumkara, Kevin T. Mellem, Zachary K. Sweeney, Elena S. Koltun, US Patent 10,882,883. 2021

74. Modular synthesis enables molecular ju-jitsu in the fight against antibiotic resistance Daniel J. Blair and Martin D. Burke Nature 2020 586, 32-33 DOI: 10.1038/d41586-020-02565-1

73. A Mild Method for Making MIDA Boronates Aidan M. Kelly, Peng-Jui Chen, Jenna Klubnick, Daniel J. Blair, and Martin D. Burke Organic Letters 2020, 22 (24), 9408-9414 DOI: 10.1021/acs.orglett.0c02449

72. Small Molecule Channels Harness Membrane Potential to Concentrate Potassium in trk1Δtrk2Δ Yeast, Jennifer Hou, Page N. Daniels, and Martin D. Burke ACS Chemical Biology2020,15 (6), 1575-1580 DOI: 10.1021/acschembio.0c00180

71. A Computer Conquers Tactical Combinations, Daniel J. Blair and Martin D. Burke Chem. 2020, 6 (1), 12-13 DOI: 10.1016/j.chempr.2019.12.019

70. Stereoretentive Cross-coupling Of Boronic Acids, Martin D. Burke, Ian Crouch, Jonathan Lehmann, Andrea Palazzolo, Claire Simons, US Patent 10,370,393. 2019

69. Amphotericin B derivatives with improved therapeutic index, Martin D. Burke, Stephen Davis, Brice E. Uno, Justin Struble, Ian Dailey, Kaitlyn C. Gray, David M. Knapp, US Patent 10,323,057. 2019

68. Modular Syntheses of Phenanthroindolizidine Natural Products Young-In Jo, Martin D. Burke, and Cheol-Hong Cheon Organic Letters2019,21 (11), 4201-4204 DOI: 10.1021/acs.orglett.9b01397

67. Axial shielding of Pd(II) complexes enables perfect stereoretention in Suzuki-Miyaura cross-coupling of Csp3 boronic acids, Jonathan W. Lehmann, Ian T. Crouch, Daniel J. Blair, Melanie Trobe, Pulin Wang, Junqi Li and Martin D. Burke Nature Communications2019,10, 1263 DOI: 10.1038/s41467-019-09249-z

66. Small-molecule ion channels increase host defences in cystic fibrosis airway epithelia. Katrina A. Muraglia, Rajeev S. Chorghade, Bo Ram Kim, Xiao Xiao Tang, Viral S. Shah, Anthony S. Grillo, Page N. Daniels, Alexander G. Cioffi, Philip H. Karp, Lingyang Zhu, Michael J. Welsh and Martin D. Burke Nature 2019, 567, 405–408 DOI: 10.1038/s41586-019-1018-5

65. FAM210B is an erythropoietin target and regulates erythroid heme synthesis by controlling mitochondrial iron import and ferrochelatase activity, Yvette Y. Yien, Jiahai Shi, Caiyong Chen, Jesmine T.M. Cheung, Anthony S. Grillo, Rishna Shrestha, Liangtao Li, Xuedi Zhang, Martin D. Kafina, Paul D. Kingsley, Matthew J. King, Julien Ablain, Hojun Li, Leonard I. Zon, James Palis, Martin D. Burke, Daniel E. Bauer, Stuart H. Orkin, Carla M. Koehler, John D. Phillips, Jerry Kaplan, Diane M. Ward, Harvey F. Lodish and Barry H. Paw Journal of Biological Chemistry2018293, 19797-19811. DOI:  10.1074/jbc.RA118.002742

64. Peridinin Is an Exceptionally Potent and Membrane-Embedded Inhibitor of Bilayer Lipid Peroxidation Hannah M.S. Haley, Adam G. Hill, Alexander I. Greenwood, Eric M. Woerly, Chad M. Rienstra, and Martin D. Burke Journal of the American Chemical Society2018,140 (45), 15227-15240 DOI: 10.1021/jacs.8b06933

63. Scalable synthesis of reduced toxicity derivative of amphotericin B, Martin D. Burke, Brice E. Uno, Souvik Rakshit, US Patent 10,087,206. 2018

62. Derivatives of amphotericin B, Martin D. Burke, Arun P. Thottumkara, Kevin T. Mellem, Zachary K. Sweeney, Elena S. Koltun, US Patent 9,957,290. 2018

61. The molecular industrial revolution: automated synthesis of small molecules, Melanie Trobe and Martin D. Burke Angewandte Chemie 2018, 57, 4192-4214 DOI: 10.1002/anie.201710482

60. Solid-State NMR of highly 13C-enriched cholesterol in lipid bilayers Lisa A. Della Ripa, Zoe A. Petros, Alexander G. Cioffi, Dennis W. Piehl, Joseph M. Courtney, Martin D. Burke and Chad M. Rienstra Methods 2018, 138-139; 47-53. DOI: 10.1016/j.ymeth.2018.01.00

59. Methods for forming protected organoboronic acids, Martin D. Burke, Graham R. Dick, David M. Knapp, Eric P. Gillis, Jenna A. Klubnick, US Patent 9,908,900. 2018

58. Towards the generalized iterative synthesis of small molecules. Jonathan W. Lehmann, Daniel J. Blair and Martin D. Burke Nature Reviews Chemistry 2018, 2, 0115 DOI: 10.1038/s41570-018-0115

57. Slow release of organoboronic acids in cross-coupling reactions, Martin D. Burke, David M. Knapp, Eric P. Gillis, US Patent 9,845,317. 2017

56. Amphotericin B derivative with reduced toxicity, Martin D. Burke, Brice E. Uno, US Patent 9,738,677. 2017

55. The Natural Productome, Andrea M. E. Palazzolo, Claire L. W. Simons, Martin D. Burke Proceedings of the National Academy of Sciences2017, 114 (22) 5564-5566; DOI: 10.1073/pnas.1706266114

54. Restored iron transport by a small molecule promotes absorption and hemoglobinization in animals Anthony S. Grillo, Anna M. SantaMaria, Martin D. Kafina, Alexander G. Cioffi, Nicholas C. Huston, Murui Han, Young Ah Seo, Yvette Y. Yien, Christopher Nardone, Archita V. Menon, James Fan, Dillon C. Svoboda, Jacob B. Anderson, John D. Hong, Bruno G. Nicolau, Kiran Subedi, Andrew A. Gewirth, Marianne Wessling-Resnick, Jonghan Kim, Barry H. Paw and Martin D. Burke Science,  2017, 356 608-615. DOI: 10.1126/science.aah3862

53. MIDA Boronates Are Hydrolysed Fast and Slow by Two Different Mechanisms Jorge A. Gonzalez, O. Maduka Ogba, Gregory F. Morehouse, Nicholas Rosson, Kendall N. Houk, Andrew G. Leach, Paul H.-Y. Cheong, Martin D. Burke and Guy C. Lloyd-Jones. Nature Chemistry 2016, 8, 1067-1075. DOI: 10.1038/nchem.2571

52. Automated synthesis of small molecules using chiral, non-racemic boronates, Martin D. Burke, Junqi Li, Eric P. Gillis, US Patent 9,388,131. 2016

51. Methods for forming protected organoboronic acids, Martin D. Burke, Graham R. Dick, David M. Knapp, Eric P. Gillis, Jenna A. Klubnick, US Patent 9,353,131. 2016

50. Slow release of organoboronic acids in cross-coupling reactions, Martin D. Burke, David M. Knapp, Eric P. Gillis, US Patent 9,328,102. 2016

49. System for controlling the reactivity of boronic acids, Martin D. Burke, Eric P. Gillis, US Patent 9,328,127. 2016

48. Our Path to Less Toxic Amphotericins, Matthew M. Endo Alexander G. Cioffi, Martin D. Burke Synlett 2015, 27, 337. DOI: 10.1055/s-0035-1560800 Recipient of the Thieme IUPAC Prize in Synthetic Organic Chemistry.

47. Apparatus and methods for the automated synthesis of small molecules, Martin D. Burke, Eric P. Gillis, Steven G. Ballmer, US Patent 9,238,597. 2016

46. C3-OH of Amphotericin B Plays an Important Role in Ion Conductance, Stephen A. Davis, Lisa A. Della Ripa, Lingbowei Hu, Alexander G. Cioffi, Taras V. Pogorelov, Chad M. Rienstra, and Martin D. Burke Journal of the American Chemical Society2015137 (48), 15102-15104 DOI: 10.1021/jacs.5b05766

45.Restored Physiology in Protein-Deficient Yeast by a Small Molecule Channel Alexander G. Cioffi, Jennifer Hou, Anthony S. Grillo, Katrina A. Diaz, and Martin D. Burke Journal of the American Chemical Society 2015 137 (32), 10096-10099 DOI: 10.1021/jacs.5b05765

44. Nontoxic Antimicrobials that Evade Drug Resistance, Stephen A. Davis, Benjamin M. Vincent, Matthew M. Endo, Luke Whitesell, Karen Marchillo, David R. Andes, Susan Lindquist and Martin D. Burke.Nature Chemical Biology 2015, 11, 481-487. DOI: 10.1038/nchembio.1821

43. Automated synthesis of small molecules using chiral, non-racemic boronates, Martin D. Burke, Junqi Li, Eric P. Gillis, US Patent 9,012,658. 2015

42. Slow release of organoboronic acids in cross-coupling reactions, Martin D. Burke, David M. Knapp, Eric P. Gillis, US Patent 9,006,463. 2015

41. Synthesis of many different types of organic small molecules using one automated process, Junqi Li, Steven G. Ballmer, Eric P. Gillis, Seiko Fujii, Michael J. Schmidt, Andrea M. E. Palazzolo, Jonathan W. Lehmann, Greg F. Morehouse, and Martin D. Burke Science 2015, 347, 1221-1226 DOI: 10.1126/science.aaa5414

40. From Synthesis to Function via Iterative Assembly of N-Methyliminodiacetic Acid Boronate Building Blocks Junqi Li, Anthony S. Grillo, and Martin D. Burke. Accounts of Chemical Research 201548 (8), 2297-2307 DOI: 10.1021/acs.accounts.5b00128

39. Cyclopropyl PIDA boronate, M Duncton, Martin D. Burke, US Patent 8,754,251. 2014

38. Synthesis of Most Polyene Natural Product Motifs Using Just Twelve Building Blocks and One Coupling Reaction, Eric M. Woerly, Jahnabi Roy, Martin D. Burke. Nature Chemistry 2014,6, 484-491.
DOI: 10.1038/nchem.1947

37. Amphotericin Forms an Extramembranous and Fungicidal Sterol Sponge, Thomas M. Anderson, Mary C. Clay, Alexander G. Cioffi, Katrina A. Diaz, Grant S. Hisao, Marcus D. Tuttle, Andrew J. Nieuwkoop, Gemma Comellas, Nashrah Maryum, Shu Wang, Brice E. Uno, Erin L. Wildeman, Tamir Gonen, Chad M. Rienstra, Martin D. Burke. Nature Chemical Biology 2014, 10, 400-406. DOI: 10.1038/nchembio.1496

36. Methods for forming protected organoboronic acids, Martin D. Burke, Graham R. Dick, David M. Knapp, Eric P. Gillis, Jenna A. Klubnick, US Patent 8,557,980. 2013

35. (1-Bromovinyl)-MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis, Eric M. Woerly, Jonathan E. Miller, and Martin D. Burke Tetrahedron 2013,69, 7732-7740. DOI: 10.1016/j.tet.2013.05.050

34. C2′-OH of Amphotericin B Plays an Important Role in Binding the Primary Sterol of Human Cells but Not Yeast Cells, Brandon C. Wilcock, Matthew M. Endo, Brice E. Uno, and Martin D. Burke Journal of the American Chemical Society2013135 (23), 8488-8491 DOI: 10.1021/ja403255s

33. Slow release of organoboronic acids in cross-coupling reactions, Martin D. Burke, David M. Knapp, Eric P. Gillis, US Patent 8,338,601. 2012

32. Electronic tuning of site-selectivity, Brandon C Wilcock 1, Brice E. Uno, Gretchen L. Bromann, Matthew J. Clark, Thomas M. Anderson and Martin D. Burke Nature Chemistry 2012, 4, 996-1003. DOI: 10.1038/nchem.1495

31. Amphotericin primarily kills yeast by simply binding ergosterol, Kaitlyn C. Gray, Daniel S. Palacios, Ian Dailey, Matthew M. Endo, Brice E. Uno, Brandon C. Wilcock, and Martin D. Burke Proceedings of the National Academy of Sciences U.S.A.2012109, 2234-223 DOI: 10.1073/pnas.1117280109

30. A General Solution for the 2-Pyridyl Problem Graham R. Dick, Eric M. Woerly and Martin D. Burke, Angewandte Chemie International Edition 2012, 51, 2667-2672 DOI: 10.1002/anie.201108608

29. Pinene-Derived Iminodiacetic Acid (PIDA): A Powerful Ligand for Stereoselective Synthesis and Iterative Cross-Coupling of C(sp3) Boronate Building Block Junqi Li and Martin D. Burke Journal of the American Chemical Society 2011,133 (35), 13774-13777 DOI: 10.1021/ja205912y

28. System for controlling the reactivity of boronic acids, Martin D. Burke, Eric P. Gillis, Suk Joong Lee, David M. Knapp, Kaitlyn C. Gray, US Patent 8,013,203. 2011

27. Total Synthesis of Synechoxanthin through Iterative Cross-Coupling, Seiko Fujii, Stephanie Y. Chang and Martin D. Burke Angewandte Chemie International Edition 2011, 50, 7862-7864. DOI: 10.1002/anie.201102688

26. Synthesis-enabled functional group deletions reveal key underpinnings of amphotericin B ion channel and antifungal activities, Daniel S. Palacios, Ian Dailey, David M. Siebert, Brandon C. Wilcock, and Martin D. Burke Proceedings of the National Academy of Sciences U.S.A. 2011, 108, 6733-6738. DOI: 10.1073/pnas.1015023108

25. (Z)-(2-Bromovinyl)-MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis, Eric M. Woerly, Justin R. Struble, Nagarjuna Palyam, Sean P. O’Hara, and Martin D. Burke Tetrahedron 2011,67, 4333-4343. DOI: 10.1016/j.tet.2011.04.021

24. A Simple and General Platform for Generating Stereochemically Complex Polyene Frameworks by Iterative Cross-Coupling Suk Joong Lee, Thomas M. Anderson, Martin D. Burke Angewandte Chemie International Edition 2010, 49, 8860-8863. DOI: 10.1002/anie.201004911

23. Stereoretentive Suzuki−Miyaura Coupling of Haloallenes Enables Fully Stereocontrolled Access to (−)-Peridinin Eric M. Woerly, Alan H. Cherney, Erin K. Davis, and Martin D. Burke Journal of the American Chemical Society 2010, 132 (20), 6941-6943 DOI: 10.1021/ja102721p

22. A General Method for Synthesis of 2-Heterocyclic N-Methyliminodiacetic Acid Boronates Graham R. Dick, David M. Knapp, Eric P. Gillis, and Martin D. Burke Organic Letters 2010, 12 (10), 2314-2317 DOI: 10.1021/ol100671v

21. N-(Carboxymethyl)-N-methyl-glycine Ian Dailey and Martin D. Burke Encyclopedia of Reagents for Organic Synthesis 2010, DOI: 10.1002/047084289X.rn01228

20. Ethynyl MIDA boronate: a readily accessible and highly versatile building block for small molecule synthesis, Graham R. Dick, David M. Knapp, Eric P. Gillis, and Martin D. Burke Tetrahedron 2010, 66, 4710-4718 DOI: 10.1016/j.tet.2010.04.020

19. A general solution for unstable boronic acids: Slow-release cross-coupling from air-stable MIDA boronates, David M. Knapp, Eric P. Gillis, Martin D. Burke Journal of the American Chemical Society, 2009 131(20), 6961-6963 DOI: 10.1021/ja901416p

18. Vinyl MIDA Boronate: a readily accessible and highly versatile building block for small molecule synthesis, Brice E. Uno, Eric P. Gillis, Martin D. Burke Tetrahedron 2009, 65, 3130-3138 DOI: 10.1016/j.tet.2010.04.020

Special Issue dedicated to Professor Justin Dubois’ receipt of the 2008 Tetrahedron Young Investigator Award

17. Flexible tetracycline synthesis yields promising antibiotics Martin D. Burke Nature Chemical Biology 2009, 5, 77-79 DOI: 10.1038/nchembio0209-77

16. B-Protected Haloboronic Acids for Iterative Cross-Coupling, Steven G. Ballmer, Eric P. Gillis, Martin D. Burke, Daniel Morton and Huw M.L. Davies Organic Syntheses 2009, 86, 344-359 DOI: 10.1002/0471264229.os086.33

15. Iterative Cross-Couplng with MIDA Boronates: Towards a General Platform for Small Molecule Synthesis, Eric P. Gillis and Martin D. Burke Aldrichimica Acta. 2009, 42(1): 17–27. DOI: 10.1002/0471264229.os086.33

14. Multistep Synthesis of Complex Boronic Acids from Simple MIDA Boronates, Eric P. Gillis and Martin D. Burke Journal of the American Chemical Society 2008, 130 (43), 14084-14085 DOI: 10.1021/ja8063759

13. Simple, Efficient, and Modular Syntheses of Polyene Natural Products via Iterative Cross-Coupling Suk Joong Lee, Kaitlyn C. Gray, James S. Paek, and Martin D. Burke Journal of the American Chemical Society 2008, 130 (2), 466-468 DOI: 10.1021/ja078129x

12. A Post-PKS Oxidation of the Amphotericin B Skeleton Predicted to be Critical for Channel Formation Is Not Required for Potent Antifungal Activity Daniel S. Palacios, Thomas M. Anderson, and Martin D. Burke Journal of the American Chemical Society 2007, 129 (45), 13804-13805 DOI: 10.1021/ja075739o

11. A Simple and Modular Strategy for Small Molecule Synthesis:  Iterative Suzuki−Miyaura Coupling of B-Protected Haloboronic Acid Building Blocks Eric P. Gillis and Martin D. Burke Journal of the American Chemical Society 2007, 129 (21), 6716-6717 DOI: 10.1021/ja0716204

10. Molecular Prosthetics: Replicating the Functions of the Molecules of Life Martin D. Burke Enhancing Chemistry Conference sponsored by the American Chemical Society. University of Illinois at Urbana-Champaign, Urbana, Illinois, March 17, 2006.

9. A Synthesis Strategy Yielding Skeletally Diverse Small Molecules Combinatorically, Martin D. Burke, Eric M. Berger, and Stuart L. Schreiber Journal of the American Chemical Society 2004 126 (43), 14095-14104 DOI: 10.1021/ja0457415

8. A planning strategy for diversity-oriented synthesis Martin D. Burke and Stuart L. Schreiber Angewandte Chemie International Edition 2004, 43, 46-58. DOI: 10.1002/anie.200300626

7. Generating Diverse Skeletons of Small Molecules Combinatorially Martin D. Burke, Eric M. Berger, and Stuart L. Schreiber Science 2003, 302, 613-618 DOI: 10.1126/science.1089946

6. Chemoenzymatic Route to Macrocyclic Hybrid Peptide/Polyketide-like Molecules Rahul M. Kohli, Martin D. Burke, Junhua Tao, and Christopher T. Walsh Journal of the American Chemical Society 2003, 125 (24), 7160-7161 DOI: 10.1021/ja0352202

5. Teaching Target-Oriented and Diversity-Oriented Organic Synthesis at Harvard University. Martin D. Burke and Gojko Lalic Chemistry and Biology 2002, 9, 535-541. DOI: 10.1016/S1074-5521(02)00143-6

4. Conformationally restricted hybrid analogues of the hormone 1 alpha,25-dihydroxyvitamin D (3): design, synthesis, and biological evaluation, M. Christina White, Martin D. Burke, Sarah Peleg, Patrick Dolan, Thomas W. Kensler, Henry Brem, and Gary H. Posner Bioorganic & Medicinal Chemistry 2001, 9, 1691-1699 DOI: 10.1016/s0968-0896(01)00087-6

3. Central Nervous System, Drug Delivery to Treat, Martin D. Burke, Henry Brem, and Robert Langer in The Encyclopedia of Controlled Drug Delivery The Encyclopedia of Controlled Drug Delivery.  Mathiowitz, E., Ed.; John Wiley and Sons., Vol. 1, 1999, 184-212.

2. Noncalcemic, Antiproliferative, Transcriptionally Active, 24-Fluorinated Hybrid Analogues of the Hormone 1α,25-Dihydroxyvitamin D3. Synthesis and Preliminary Biological Evaluation Gary H. Posner, Jae Kyoo Lee, Qiang Wang, Sara Peleg, Martin D. Burke, Henry Brem, Patrick Dolan, and Thomas W. Kensler Journal of Medicinal Chemistry 1998, 41 (16), 3008-3014 DOI: 10.1021/jm980031t

1.Polymer-Controlled Drug Delivery: An Overview for the Clinician, Justin Hanes and Martin D. Burke.  Hospital Pharmacist Report.  December 1997 2-11